Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Methylated-DNA--protein-cysteine methyltransferase' and Ligand = 'BDBM5484'
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM5484(6-(cyclopent-1-en-1-ylmethoxy)-9H-purin-2-amine | ...)
Affinity DataIC50:  200nMAssay Description:concentration required to reduce AGT activity to 50% of control rate in intact HT-29 human colorectal carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM5484(6-(cyclopent-1-en-1-ylmethoxy)-9H-purin-2-amine | ...)
Affinity DataIC50:  390nMAssay Description:Inhibition of AGT activity to 50% of control rate in HT-29 cell extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed