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Found 4 Enz. Inhib. hit(s) with Target = 'Motilin receptor' and Ligand = 'BDBM50199365'
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199365((E)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl...)
Affinity DataKi:  137nMAssay Description:Displacement of [125I]-motilin from human motilin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199365((E)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl...)
Affinity DataKi:  137nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199365((E)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl...)
Affinity DataIC50:  74nMAssay Description:Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199365((E)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl...)
Affinity DataIC50:  74nMAssay Description:Activity at human MOTR expressed in CHO cells assessed as inhibition of motilin-induced calcium releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed