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Found 2 Enz. Inhib. hit(s) with Target = 'Motilin receptor' and Ligand = 'BDBM50214262'
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50214262((5R,8R,11S)-5-[(4-chlorophenyl)methyl]-11-[(methyl...)
Affinity DataKi:  31nMAssay Description:Displacement of [125I]-motilin from human motilin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMotilin receptor(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50214262((5R,8R,11S)-5-[(4-chlorophenyl)methyl]-11-[(methyl...)
Affinity DataIC50:  33nMAssay Description:Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed