TargetMotilin receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:In vitro binding affinity towards human motilin receptorMore data for this Ligand-Target Pair
TargetMotilin receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataEC50: 4.20nMAssay Description:In vitro effective concentration towards human motilin receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as increase of muscle contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair