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Found 8 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM224024'
TargetMu-type opioid receptor(GUINEA PIG)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataKi:  0.920nMAssay Description:Binding affinity to Opioid receptor mu 1 by competitive inhibition of radioligand [3H]-DAMGO using cloned receptors transiently expressed on CHO cell...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Sri International

Curated by PDSP Ki Database
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataKi:  4.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataKi:  50nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of mu-selective antagonist binding to opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Oregon State University

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of [3H]-PL-17 binding to mu opioid receptor of guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Sri International

Curated by PDSP Ki Database
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataEC50:  214nMAssay Description:Agonist activity at human recombinant MOR expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Sri International

Curated by PDSP Ki Database
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataEC50:  214nMAssay Description:Agonist activity at human recombinant MOR expressed in CHO cells assessed as calcium mobilization by Fluo-4 AM based fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed