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Found 8 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50068664'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  1.72E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  1.72E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  3.22E+3nMAssay Description:Tested for binding affinity against mu opioid receptor fby displacing [3H]- DAMGO radioligand from rat brain membrane preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  3.23E+3nMAssay Description:Tested for binding affinity against mu opioid receptor fby displacing [3H]- DAMGO radioligand from rat brain membrane preparationsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi: >4.50E+3nMAssay Description:Affinity towards human Opioid receptor mu 1 on CHO cell membranes using [3H]DAMGO displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 on rat forebrain membranes by [3H]sufentanil displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50068664(2-[2-({(S)-2-[2-Amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as effect on muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed