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Found 2 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50237596'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Medical University Of Lodz

Curated by ChEMBL
LigandPNGBDBM50237596(CHEMBL4099423)
Affinity DataKi:  0.730nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain homogenates after 180 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Medical University Of Lodz

Curated by ChEMBL
LigandPNGBDBM50237596(CHEMBL4099423)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant MOR expressed in CHO cells assessed as calcium mobilization by Fluo-4 AM based fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed