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Found 5 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50453048'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453048(CHEMBL2115042)
Affinity DataKi:  1.70E+3nMAssay Description:Binding affinity measured against [3H]CTOP (Opioid receptor mu 1) in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453048(CHEMBL2115042)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibitory activity measured against [3H]CTOP binding to Opioid receptor mu 1 in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453048(CHEMBL2115042)
Affinity DataIC50:  4.83E+4nMAssay Description:Inhibitory activity measured against Opioid receptor mu 1 using guinea pig ileum assay (GPI).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453048(CHEMBL2115042)
Affinity DataIC50:  6.90E+4nMAssay Description:Binding affinity measured against [3H]CTOP binding to Opioid receptor mu 1 in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453048(CHEMBL2115042)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibitory activity measured against [3H]CTOP (Opioid receptor mu 1) in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed