Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity measured against [3H]CTOP (Opioid receptor mu 1) in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Inhibitory activity measured against [3H]CTOP binding to Opioid receptor mu 1 in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: 4.83E+4nMAssay Description:Inhibitory activity measured against Opioid receptor mu 1 using guinea pig ileum assay (GPI).More data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+4nMAssay Description:Binding affinity measured against [3H]CTOP binding to Opioid receptor mu 1 in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibitory activity measured against [3H]CTOP (Opioid receptor mu 1) in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair