Affinity DataKi: 24nMAssay Description:Binding affinity measured against [3H]CTOP (Opioid receptor mu 1) in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Inhibitory activity measured against [3H]CTOP (Opioid receptor mu 1) in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity measured against Opioid receptor mu 1 using guinea pig ileum assay (GPI).More data for this Ligand-Target Pair