Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM83396'
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM83396(1-(4-acetamidobenzyl)-4-phenethyl-isonipecotic aci...)
Affinity DataEC50:  8.30E+3nMAssay Description:Inhibition of mu opioid receptor (unknown origin) expressed in human UO5S cells assessed as increase in beta arrestin recruitmentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM83396(1-(4-acetamidobenzyl)-4-phenethyl-isonipecotic aci...)
Affinity DataEC50:  945nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM83396(1-(4-acetamidobenzyl)-4-phenethyl-isonipecotic aci...)
Affinity DataEC50:  125nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM83396(1-(4-acetamidobenzyl)-4-phenethyl-isonipecotic aci...)
Affinity DataEC50:  54nMAssay Description:Inhibition of mu opioid receptor (unknown origin) expressed in human UO5S cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed