Found 5 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1' and Ligand = 'BDBM50305083' TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of MRP1More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataIC50: 6.65E+3nMAssay Description:Inhibition of human ABCC1 transfected in MDCK2-MRP1 cells using calcein-AM as substrate measured after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataIC50: >8.00E+3nMAssay Description:Inhibition of ABCC1 mediated etoposide resistant in human 2008 cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataEC50: 1.95E+3nMAssay Description:Inhibition of MRP1 (unknown origin) expressed in human 2008/MRP1 assessed as reversal of doxorubicin resistance after 5 days by MTS/PMS assayMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Inhibition of MRP1 (unknown origin) expressed in human 2008/MRP1 cells assessed as potentiation of mitoxantrone-induced cytotoxicity after 5 days by ...More data for this Ligand-Target Pair
