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Found 1 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1' and Ligand = 'BDBM50344959'
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Queen'S University

Curated by ChEMBL
LigandPNGBDBM50344959(17beta-Estradiol-17-(beta-D-glucuronide) | CHEMBL1...)
Affinity DataKi:  2.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed