Found 6 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1/M2/M3/M4/M5' and Ligand = 'BDBM21398'
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Prestwick Chemical
Curated by ChEMBL
Prestwick Chemical
Curated by ChEMBL
Affinity DataKi: 4.67E+3nMAssay Description:Binding affinity towards human muscarinic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.47E+3nMAssay Description:In vitro binding affinity against Muscarinic acetylcholine receptors in rat brain.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition the uptake of tritiated serotonin (5-HT) by the serotonin transporter SERT in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:The compound was tested for inhibition of [3H]QNB binding to Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60E+3nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor in rat brain using [3H]- QNBMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:The ability to displace [3H]QNB from Muscarinic acetylcholine receptor in rat brain membrane was determinedMore data for this Ligand-Target Pair