Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50107696'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo
Curated by ChEMBL
The University Of Toledo
Curated by ChEMBL
Affinity DataKi: 0.840nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo
Curated by ChEMBL
The University Of Toledo
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]NMS from human M1 receptor expressed in CHO cells by microplate scintillation counting based radioligand binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo
Curated by ChEMBL
The University Of Toledo
Curated by ChEMBL
Affinity DataEC50: 720nMAssay Description:Agonistic activity against M1 muscarinic receptor expressed in A9 L cells.More data for this Ligand-Target Pair