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Found 5 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50258439'
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50258439(1-(4-bromobenzyl)indoline-2,3-dione | CHEMBL523685...)
Affinity DataEC50:  6.04E+3nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50258439(1-(4-bromobenzyl)indoline-2,3-dione | CHEMBL523685...)
Affinity DataEC50:  6.04E+3nMAssay Description:Activation of rat muscarinic M1 receptor expressed in CHO cells coexpressing Gq protein assessed as potentiation of acetylcholine-induced intracellul...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258439(1-(4-bromobenzyl)indoline-2,3-dione | CHEMBL523685...)
Affinity DataEC50:  6.00E+3nMAssay Description:Positive allosteric modulation activity at muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258439(1-(4-bromobenzyl)indoline-2,3-dione | CHEMBL523685...)
Affinity DataEC50:  6.10E+3nMAssay Description:Positive allosteric modulation of muscarinic M1 receptor expressed in CHO cells assessed as effect on acetylcholine-induced intracellular calcium mob...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50258439(1-(4-bromobenzyl)indoline-2,3-dione | CHEMBL523685...)
Affinity DataEC50:  6.10E+3nMAssay Description:Agonist activity at rat muscarinic M1 expressed in CHO cells assessed as stimulation of calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed