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Found 5 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM73209'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM73209((+)-CIS-DIOXOLANE | CHEMBL105457 | MLS000069362 | ...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM73209((+)-CIS-DIOXOLANE | CHEMBL105457 | MLS000069362 | ...)
Affinity DataKi:  6.40nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM73209((+)-CIS-DIOXOLANE | CHEMBL105457 | MLS000069362 | ...)
Affinity DataKi:  2.10E+3nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -pirenzepine providing a measure of muscarinic m1 receptor antagonist affinityMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM73209((+)-CIS-DIOXOLANE | CHEMBL105457 | MLS000069362 | ...)
Affinity DataKi:  1.10E+4nMAssay Description:Binding affinity to human cloned muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM73209((+)-CIS-DIOXOLANE | CHEMBL105457 | MLS000069362 | ...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor transfected in CHO cells after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed