Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM50268343'
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50268343(CHEMBL4096727)
Affinity DataIC50:  427nMAssay Description:Antagonist activity at human muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50268343(CHEMBL4096727)
Affinity DataIC50:  440nMAssay Description:Antagonist activity at human recombinant muscarinic M4 receptor expressed in CHO cells co-transfected with Gqi5 in presence of EC80 acetylcholine by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50268343(CHEMBL4096727)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed