Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M5' and Ligand = 'BDBM50023229'
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt University Medical Center
Curated by ChEMBL
Vanderbilt University Medical Center
Curated by ChEMBL
Affinity DataEC50: 610nMAssay Description:Activity at rat muscarinic acetylcholine receptor subtype 5 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Positive allosteric modulation of M5 AchR (unknown origin) assessed as increase in acetylcholine-induced responseMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Positive allosteric modulator activity at human muscarinic acetylcholine receptor subtype 5 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 195nMAssay Description:Positive allosteric modulator activity at human muscarinic acetylcholine receptor subtype 5 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair