Found 4 Enz. Inhib. hit(s) with Target = 'N-terminal Xaa-Pro-Lys N-methyltransferase 1' and Ligand = 'BDBM50553069'
Affinity DataIC50: 340nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged NTMT1 (1 to 222 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using GPKRIA p...More data for this Ligand-Target Pair
Affinity DataIC50: 4.38E+3nMAssay Description:Inhibition of NTMT1 (unknown origin) using SPKRIAKRRS(CONH2) peptide as substrate assessed as SAH production incubated for 10 mins in the presence of...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of NTMT1 in human HT29 cells assessed as decrease in me3-RCC1 level incubated for 3 days by Western blot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of NTMT1 in human HCT116 cells assessed as decrease in me3-RCC1 level incubated for 3 days by Western blot analysisMore data for this Ligand-Target Pair