Found 2 Enz. Inhib. hit(s) with Target = 'NAD-dependent protein deacetylase sirtuin-1' and Ligand = 'BDBM50576687'
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
The University Of Hong Kong
Curated by ChEMBL
The University Of Hong Kong
Curated by ChEMBL
Affinity DataKi: 4.80E+4nMAssay Description:Inhibition of human recombinant SIRT1 assessed as inhibition of substrate deacetylation using Gln-Pro-Lys-Lys- (epsilon acetyl) AMC peptide as substr...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
The University Of Hong Kong
Curated by ChEMBL
The University Of Hong Kong
Curated by ChEMBL
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of human recombinant SIRT1 assessed as inhibition of substrate deacetylation using Gln-Pro-Lys-Lys- (epsilon acetyl) AMC peptide as substr...More data for this Ligand-Target Pair