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Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-3/beta-4' and Ligand = 'BDBM50331014'
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Sri International

Curated by ChEMBL
LigandPNGBDBM50331014(9-methyl-3-(pyridin-3-yl)-9-azabicyclo[3.3.1]non-2...)
Affinity DataKi:  241nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK292 cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Sri International

Curated by ChEMBL
LigandPNGBDBM50331014(9-methyl-3-(pyridin-3-yl)-9-azabicyclo[3.3.1]non-2...)
Affinity DataEC50:  4.80E+3nMAssay Description:Partial agonist activity at rat alpha3beta4 nAChR expressed in HEK292 cells assessed as increase of calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed