Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4' and Ligand = 'BDBM50088432'
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50088432(5-(1,4-diazepan-1-yl)nicotinamide | 5-[1,4]Diazepa...)
Affinity DataIC50:  19.9nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
University Of Turin

Curated by ChEMBL
LigandPNGBDBM50088432(5-(1,4-diazepan-1-yl)nicotinamide | 5-[1,4]Diazepa...)
Affinity DataEC50:  1.29E+4nMAssay Description:Agonist activity at human alpha4beta2 nAChR expressed in HEK293 cells assessed as intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed