Found 8 Enz. Inhib. hit(s) with Target = 'Non-lysosomal glucosylceramidase' and Ligand = 'BDBM18355'
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
University Of Napoli Federico Ii
Curated by ChEMBL
University Of Napoli Federico Ii
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of NLGase in human SH-SY5Y cells using MUG-Gluc as fluorogenic substrate preincubated for 30 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of conduritol beta-epoxide-sensitive mouse glucosylceramidaseMore data for this Ligand-Target Pair
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
University Of Napoli Federico Ii
Curated by ChEMBL
University Of Napoli Federico Ii
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of recombinant GBA2 preincuabated with compound for 30 mins using 4-methylumbelliferyl-B-glucoside substrate by fluorimetric assayMore data for this Ligand-Target Pair
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
University Of Napoli Federico Ii
Curated by ChEMBL
University Of Napoli Federico Ii
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of human GBA2More data for this Ligand-Target Pair
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
University Of Napoli Federico Ii
Curated by ChEMBL
University Of Napoli Federico Ii
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of GBA2 (unknown origin)More data for this Ligand-Target Pair
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
University Of Napoli Federico Ii
Curated by ChEMBL
University Of Napoli Federico Ii
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of GBA2 by HPLCMore data for this Ligand-Target Pair
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
University Of Napoli Federico Ii
Curated by ChEMBL
University Of Napoli Federico Ii
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of glucosylceramidase 2 from spleen of patient with gaucher's disease by fluorimetric analysisMore data for this Ligand-Target Pair
TargetNon-lysosomal glucosylceramidase(Homo sapiens (Human))
University Of Napoli Federico Ii
Curated by ChEMBL
University Of Napoli Federico Ii
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of non-lysosomal glucosylceramidase in cultured melanoma cellsMore data for this Ligand-Target Pair