Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma' and Ligand = 'BDBM50044245'
TargetNuclear receptor ROR-gamma(Mus musculus)
Genentech

Curated by ChEMBL
LigandPNGBDBM50044245(CHEMBL3314043)
Affinity DataEC50: <100nMAssay Description:Activity at RoRc in mouse CD4+ T cells assessed as inhibition of IL-17 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50044245(CHEMBL3314043)
Affinity DataEC50: <100nMAssay Description:Inverse agonist activity at human RoRc-LBD expressed in cells assessed as TRAP-220 coactivator peptide recruitmentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed