Affinity DataEC50: 126nMAssay Description:Agonist activity at human ROR-gamma LBD expressed in HEK293 cells assessed as transcriptional activity in presence of ursolic acid by Gal4-luciferase...More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair