Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma' and Ligand = 'BDBM50577440'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577440(CHEMBL4870074)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human ROR-gamma LBD expressed in HEK293 cells assessed as transcriptional activity in presence of ursolic acid by Gal4-luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577440(CHEMBL4870074)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed