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Found 1 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group I member 2' and Ligand = 'BDBM23451'
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM23451(5,14-dihydroxy-8,17-dioxatetracyclo[8.7.0.0^{2,7}....)
Affinity DataIC50:  1.20E+4nMAssay Description:Antagonist activity at human PXR transfected in African green monkey CV1 cells assessed as inhibition of SR12813-induced transactivation after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed