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Found 3 Enz. Inhib. hit(s) with Target = 'Oxoeicosanoid receptor 1' and Ligand = 'BDBM50024458'
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Florida Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50024458(5-oxo-ETE | CHEMBL18028 | ETE-5-Oxo)
Affinity DataIC50:  3nMAssay Description:Desensitization of 5-oxo-ETE receptor in indo-1-labeled human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Florida Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50024458(5-oxo-ETE | CHEMBL18028 | ETE-5-Oxo)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Florida Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50024458(5-oxo-ETE | CHEMBL18028 | ETE-5-Oxo)
Affinity DataEC50:  7nMAssay Description:Agonist activity at 5-oxo-ETE receptor in human neutrophils assessed as stimulation of ca2+ mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed