Found 21 Enz. Inhib. hit(s) with Target = 'Oxytocin receptor' and Ligand = 'BDBM50139178' 
Affinity DataKi: 31nMAssay Description:Displacement of DY647 from SNAP-tagged OTR receptor (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Displacement of [Tyrosyl-2,6-3H]Oxytocin from recombinant mouse OTR expressed in CHO-K1 cells after 180 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [Tyrosyl-2,6-3H]oxytocin from recombinant human OTR expressed in CHO-DUKX-A2 cells incubated for 180 mins by scintillation counting b...More data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [3H]-vasopressin from human vasopressin 1a receptor expressed in HEK293 cells after 90 mins by microbeta 2 microplate-reader methodMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [Tyrosyl-2,6-3H]Oxytocin from recombinant human OTR expressed in CHO-DUKX-A2 cells after 180 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Displacement of [3H]-oxytocin from human OTR expressed in HEK293 cell membranes after 90 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Agonist activity at human oxytocin receptor expressed in HEK293 cells assessed as increase in IP1 accumulation preincubated for 1 hr followed by addi...More data for this Ligand-Target Pair
Affinity DataKi: 978nMAssay Description:Displacement of [tyrosyl-2,6-3H] oxytocin from OTR (unknown origin) expressed in HEK293 cell membranes incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human oxytocin receptor expressed in HEK293 cells assessed as inhibition of oxytocin induced IP1 accumulation pretreated for 3...More data for this Ligand-Target Pair
Affinity DataEC50: 78nMAssay Description:Agonist activity at mouse OTR receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Agonist activity at recombinant mouse OTR expressed in CHO-K1 cells assessed as induction of Ca2+ mobilization after overnight incubation by FLIPR as...More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at human OTR expressed in HEK cells assessed as increase in intracellular calcium flux incubated for 45 mins by Indo1-AM dye based f...More data for this Ligand-Target Pair
Affinity DataEC50: 881nMAssay Description:Agonist activity at human OTR stably expressed in HEK cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293FT cells incubated for 30 mins by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
Affinity DataEC50: 61nMAssay Description:Agonist activity at recombinant human OTR expressed in CHO-DUKX-A2 cells assessed as stimulation of intracellular calcium concentration by calcium 3 ...More data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Agonist activity at human OTR receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 420nMAssay Description:Agonist activity at human OTR expressed in HEK293 cells assessed as induction of IP1 accumulation after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 880nMAssay Description:Agonist activity at C-terminal GFP-tagged OTR (unknown origin) expressed in HEK293 cells measured after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 420nMAssay Description:Displacement of [3H]-oxytocin from human oxytocin receptor expressed in HEK293 cells after 90 mins by microbeta 2 microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 61nMAssay Description:Agonist activity at recombinant human OTR expressed in CHO-K1 cells assessed as induction of Ca2+ mobilization after overnight incubation by FLIPR as...More data for this Ligand-Target Pair
Affinity DataEC50: 61nMAssay Description:Antagonist activity at human oxytocin receptor expressed in HEK293 cells assessed as inhibition of oxytocin induced IP1 accumulation pretreated for 3...More data for this Ligand-Target Pair
