Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'P2X purinoceptor 4' and Ligand = 'BDBM50446069'
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50446069(CHEMBL3103372)
Affinity DataIC50:  3.41E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50446069(CHEMBL3103372)
Affinity DataIC50:  6.93E+4nMAssay Description:Antagonist activity at rat P2X4 receptor assessed as inhibition of ATP-induced calcium influx preincubated for 30 mins followed by ATP addition by Fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50446069(CHEMBL3103372)
Affinity DataIC50:  1.23E+5nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed