Affinity DataIC50: 10nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced ethidium uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human P2X7R transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human P2X7R transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20E+4nMAssay Description:Antagonist activity at human P2X7R transfected in HEK293 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by YOPRO-...More data for this Ligand-Target Pair
Affinity DataIC50: 9.20E+4nMAssay Description:Antagonist activity at human P2X7R transfected in HEK293 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by YOPRO-...More data for this Ligand-Target Pair