Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by turbidimetric methodMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:The compound was evaluated for antagonist activity against platelet P2Y purinoceptor 12 (P2Y12)More data for this Ligand-Target Pair
Affinity DataKd: 4.57nMAssay Description:Binding affinity to P2Y12 receptor expressed in human platelets from 0.047 to 50 nMMore data for this Ligand-Target Pair