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Found 3 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 12' and Ligand = 'BDBM50167271'
TargetP2Y purinoceptor 12(Homo sapiens (Human))TBA
LigandPNGBDBM50167271(CHEMBL3798413)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-2-MeS-ADP from human P2Y12 assessed as inhibition constant incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))TBA
LigandPNGBDBM50167271(CHEMBL3798413)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]-2-Mes-ADP from human P2Y12 receptor by beta-counter analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))TBA
LigandPNGBDBM50167271(CHEMBL3798413)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at P2Y12 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed