Affinity DataKi: 0.380nMAssay Description:Binding affinity at human recombinant P2Y12 receptor expressed in CHO cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:Inhibition of human P2Y12 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet rich plasma assessed as inhibition of ADP-induced platelet aggregation by light transmission ...More data for this Ligand-Target Pair