Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50299116'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50299116(CHEMBL574606 | rac-2-(4-Phenylethynyl-phenoxy)-3-p...)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed