Found 4 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor delta' and Ligand = 'BDBM50180197'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Sahmyook University
Curated by ChEMBL
Sahmyook University
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Sahmyook University
Curated by ChEMBL
Sahmyook University
Curated by ChEMBL
Affinity DataEC50: 1.67E+4nMAssay Description:Antagonist activity at PPARdelta LBD (unknown origin) assessed as increase in recruitment of SMRT ID2 corepressor peptide by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Sahmyook University
Curated by ChEMBL
Sahmyook University
Curated by ChEMBL
Affinity DataEC50: 1.07E+4nMAssay Description:Antagonist at PPARdelta LBD (unknown origin) assessed as increase in recruitment of coactivator peptide C33 cotreated with PPARdelta agonist GW501516...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Sahmyook University
Curated by ChEMBL
Sahmyook University
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Competitive binding affinity to GST-tagged human PPARdelta LBD incubated for 1 to 6 hrs by TR-FRET assayMore data for this Ligand-Target Pair