Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM21221'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Sahmyook University
Curated by ChEMBL
Sahmyook University
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARgamma LBD by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Sahmyook University
Curated by ChEMBL
Sahmyook University
Curated by ChEMBL
Affinity DataEC50: 2.94E+3nMAssay Description:Competitive binding affinity to GST-tagged human PPARgamma LBD incubated for 1 to 6 hrs by TR-FRET assayMore data for this Ligand-Target Pair