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Found 9 Enz. Inhib. hit(s) with Target = 'Phosphotransferase' and Ligand = 'BDBM50180152'
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas

Curated by ChEMBL
LigandPNGBDBM50180152((9-ethyl-9H-3-carbazolyl)-aminomethylene-1,1-bisph...)
Affinity DataKi:  500nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas

Curated by ChEMBL
LigandPNGBDBM50180152((9-ethyl-9H-3-carbazolyl)-aminomethylene-1,1-bisph...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas

Curated by ChEMBL
LigandPNGBDBM50180152((9-ethyl-9H-3-carbazolyl)-aminomethylene-1,1-bisph...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas

Curated by ChEMBL
LigandPNGBDBM50180152((9-ethyl-9H-3-carbazolyl)-aminomethylene-1,1-bisph...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas

Curated by ChEMBL
LigandPNGBDBM50180152((9-ethyl-9H-3-carbazolyl)-aminomethylene-1,1-bisph...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas

Curated by ChEMBL
LigandPNGBDBM50180152((9-ethyl-9H-3-carbazolyl)-aminomethylene-1,1-bisph...)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas

Curated by ChEMBL
LigandPNGBDBM50180152((9-ethyl-9H-3-carbazolyl)-aminomethylene-1,1-bisph...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas

Curated by ChEMBL
LigandPNGBDBM50180152((9-ethyl-9H-3-carbazolyl)-aminomethylene-1,1-bisph...)
Affinity DataIC50:  810nMAssay Description:Inhibition of Trypanosoma cruzi hexokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas

Curated by ChEMBL
LigandPNGBDBM50180152((9-ethyl-9H-3-carbazolyl)-aminomethylene-1,1-bisph...)
Affinity DataIC50:  810nMAssay Description:Inhibitory activity against Trypanosoma cruzi hexokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed