Found 11 Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50005232'
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Rhone-Poulenc Sante
Curated by PDSP Ki Database
Rhone-Poulenc Sante
Curated by PDSP Ki Database
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Rhone-Poulenc Sante
Curated by PDSP Ki Database
Rhone-Poulenc Sante
Curated by PDSP Ki Database
Affinity DataKi: 7.20nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory activity expressed as the concentration required to inhibit platelet-activating factor (PAF) induced maximum aggregation by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of PAF-induced platelet aggregation in rabbit platelet rich plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of rabbit platelet aggregation induced by platelet activating factor (PAF)More data for this Ligand-Target Pair