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Found 2 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase tankyrase-2' and Ligand = 'BDBM50232346'
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Health & Science University

Curated by ChEMBL
LigandPNGBDBM50232346(CHEMBL4101890)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant human TNKS2 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins followed by biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Health & Science University

Curated by ChEMBL
LigandPNGBDBM50232346(CHEMBL4101890)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant human TNKS2 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins followed by biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed