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Found 3 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily A member 3' and Ligand = 'BDBM50125521'
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50125521(CHEMBL16804 | Propyl-carbamic acid 4-[(2-methoxy-b...)
Affinity DataIC50:  5nMAssay Description:Inhibition of DiTc binding to Kv1.3 channel in human brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50125521(CHEMBL16804 | Propyl-carbamic acid 4-[(2-methoxy-b...)
Affinity DataIC50:  50nMAssay Description:Inhibition of [86Rb+] efflux from CHO cells stably transfected with Kv1.3 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50125521(CHEMBL16804 | Propyl-carbamic acid 4-[(2-methoxy-b...)
Affinity DataIC50:  273nMAssay Description:Inhibition of T-cell proliferation was determined by a human T-cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed