Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily H member 2' and Ligand = 'BDBM50395398'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395398(CHEMBL2165064)
Affinity DataIC50: >2.00E+5nMAssay Description:Displacement of [3H]-astemizole from human ERG expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395398(CHEMBL2165064)
Affinity DataIC50:  2.33E+5nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395398(CHEMBL2165064)
Affinity DataIC50:  2.33E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed