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Found 3 Enz. Inhib. hit(s) with Target = 'Prokineticin receptor 1' and Ligand = 'BDBM121157'
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents of The University of California

US Patent
LigandPNGBDBM121157(US8722896, (+/-)-2-Methyl-3-(2,3-dihydro-1- benzof...)
Affinity DataKi:  3.78nM ΔG°:  -50.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents of The University of California

US Patent
LigandPNGBDBM121157(US8722896, (+/-)-2-Methyl-3-(2,3-dihydro-1- benzof...)
Affinity DataKi:  7.44nM ΔG°:  -48.3kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents of The University of California

US Patent
LigandPNGBDBM121157(US8722896, (+/-)-2-Methyl-3-(2,3-dihydro-1- benzof...)
Affinity DataKi:  13.6nM ΔG°:  -46.7kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails US Patent