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Found 3 Enz. Inhib. hit(s) with Target = 'Prolyl endopeptidase' and Ligand = 'BDBM554517'
TargetProlyl endopeptidase(Homo sapiens (Human))
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM554517((5RS)—N-Cyclopropyl-2-(4-methylbenzyl)-3-oxo-...)
Affinity DataIC50:  0.325nMAssay Description:To recombinant full-length human prolyl endopeptidase (PREP, R&D-Systems, 4308-SE; final concentration, for example, 0.4 nM, volume: 25 al) in reacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM554517((5RS)—N-Cyclopropyl-2-(4-methylbenzyl)-3-oxo-...)
Affinity DataIC50:  0.350nMAssay Description:To recombinant full-length human prolyl endopeptidase (PREP, R&D-Systems, 4308-SE; final concentration, for example, 0.4 nM, volume: 25 al) in reacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Bayer Aktiengesellschaft

US Patent
LigandPNGBDBM554517((5RS)—N-Cyclopropyl-2-(4-methylbenzyl)-3-oxo-...)
Affinity DataIC50:  120nMAssay Description:To recombinant full-length human prolyl endopeptidase (PREP, R&D-Systems, 4308-SE; final concentration, for example, 0.4 nM, volume: 25 al) in reacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent