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Found 2 Enz. Inhib. hit(s) with Target = 'Prolyl hydroxylase EGLN2' and Ligand = 'BDBM50239937'
TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50239937(CHEMBL4083851 | US10287286, Example 3)
Affinity DataIC50:  34nMAssay Description:Inhibition of full length HIF-PHD1 (unknown origin) expressed in baculovirus infected sf9 cells using DLDLEMLAPYIPMDDDFQL/2-Oxoglutarate as substrate...More data for this Ligand-Target Pair
TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50239937(CHEMBL4083851 | US10287286, Example 3)
Affinity DataIC50:  34nMAssay Description:The IC50 values for the PHD1 enzyme (residues 1-407) were determined by mixing increasing amounts of a compound of the invention with a fixed amount ...More data for this Ligand-Target Pair