Found 1 Enz. Inhib. hit(s) with Target = 'Proprotein convertase subtilisin/kexin type 7' and Ligand = 'BDBM50349829'
TargetProprotein convertase subtilisin/kexin type 7(Homo sapiens (Human))
Universidade Estadual Paulista
Curated by ChEMBL
Universidade Estadual Paulista
Curated by ChEMBL
Affinity DataIC50: 462nMAssay Description:Inhibition of recombinant type 8 subtilisin using Arg-Glu-(EDANS)- Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Lys-(DALBCYL)-Arg fluorogenic substrate preincubat...More data for this Ligand-Target Pair