Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-5' and Ligand = 'BDBM50518157'
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518157(CHEMBL4522493)
Affinity DataKi:  4.80nMAssay Description:Non-competitive mixed-type inhibition of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518157(CHEMBL4522493)
Affinity DataIC50:  50nMAssay Description:Negative allosteric modulation of SDS-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518157(CHEMBL4522493)
Affinity DataIC50:  500nMAssay Description:Negative allosteric modulation of 10 uM Rpt5-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50518157(CHEMBL4522493)
Affinity DataIC50:  560nMAssay Description:Negative allosteric modulation of 1 uM Rpt5-activated human erythrocytes 20S proteasome chymotrypsin like activity using Suc-LLVY-AMC as substrate me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed