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Found 3 Enz. Inhib. hit(s) with Target = 'Protein ENL' and Ligand = 'BDBM50466617'
TargetProtein ENL(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466617(CHEMBL4287247)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by alphascreen ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtein ENL(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466617(CHEMBL4287247)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to recombinant C-terminal His6-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in expressed Escherichia coli ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtein ENL(Homo sapiens)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50466617(CHEMBL4287247)
Affinity DataKd:  6.10E+3nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB