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Found 1 Enz. Inhib. hit(s) with Target = 'Protein arginine N-methyltransferase 8' and Ligand = 'BDBM50158097'
TargetProtein arginine N-methyltransferase 8(Homo sapiens (Human))
University Of Toronto

Curated by ChEMBL
LigandPNGBDBM50158097(CHEMBL3780701)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human PRMT8 using 24 residues of biotin labelled histone4 substrate and tritiated 3H-S-adenosylmethionine by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed