Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM13316'
LigandPNGBDBM13316(1-Methyl-1H-imidazole-4-sulfonic Acid Biphenyl-4-y...)
Affinity DataIC50:  880nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed