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Found 6 Enz. Inhib. hit(s) with Target = 'Protein kinase C gamma type' and Ligand = 'BDBM3152'
TargetProtein kinase C gamma type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Protein kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C gamma type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  12nMAssay Description:Inhibition of protein kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C gamma type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  12nMAssay Description:Inhibition of protein kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C gamma type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Protein Kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C gamma type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  13nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C gamma isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  13nMpH: 7.5 T: 2°CAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails Article